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Hexarelin

Also known as: Examorelin

Growth HormonePHASE 2

Clinical Status

Investigational — clinical trials conducted.

Mechanism of Action

Activates ghrelin receptors causing potent GH release. Uniquely binds to CD36 receptors in cardiac tissue, providing cardioprotective effects independent of GH.

Dosing Defaults

Dose

100-200 mcg

Frequency

2-3x daily

Administration

Subcutaneous injection

Timing

Morning and before bed (fasted)

Food

fasted

Duration

4-8 weeks

Dose range: 100-300 mcg per dose

Take fasted for maximum GH response.

Side Effects

  • Increased appetite
  • Water retention
  • Tingling/numbness
  • Elevated cortisol and prolactin
  • Flushing
  • Receptor desensitization with continuous use

Contraindications & Warnings

  • Active malignancy
  • Not medical advice
  • Desensitization occurs with continuous use — cycle off

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This information is for educational purposes only and is not medical advice. Dosing data is based on research literature and community reports. Always consult a qualified healthcare provider before using any peptide.